EC 2.7.11.2 - ATP:[pyruvate dehydrogenase (acetyl- transferring) ] phosphotransferase ([pyruvate dehydrogenase (acetyl- transferring) ] kinase)

3D structures of EC 2.7.11.2 - [pyruvate dehydrogenase (acetyl-transferring)] kinase in Protein Data Bank

updated: 6 January 2022, 2:15

1. 3d2r: Crystal Structure of Pyruvate Dehydrogenase Kinase Isoform 4 in Complex with Adp
2. 3crl: Crystal Structure of The Pdhk2-l2 Complex.
3. 3crk: Crystal Structure of The Pdhk2-l2 Complex.
4. 2zkj: Crystal Structure of Human Pdk4-adp Complex
5. 2zdy: Inhibitor-bound Structures of Human Pyruvate Dehydrogenase Kinase 4
6. 2zdx: Inhibitor-bound Structures of Human Pyruvate Dehydrogenase Kinase 4
7. 2q8i: Pyruvate Dehydrogenase Kinase Isoform 3 in Complex with Antitumor Drug Radicicol
8. 2q8h: Structure of Pyruvate Dehydrogenase Kinase Isoform 1 in Complex with Dichloroacetate (dca)
9. 2q8g: Structure of Pyruvate Dehydrogenase Kinase Isoform 1 in Complex with Glucose-lowering Drug Azd7545
10. 2q8f: Structure of Pyruvate Dehydrogenase Kinase Isoform 1
11. 2pnr: Crystal Structure of The Asymmetric Pdk3-l2 Complex
12. 2e0a: Crystal Structure of Human Pyruvate Dehydrogenase Kinase 4 in Complex with Amppnp
13. 6lio: Crystal Structure of Human Pdk2 Complexed with Gm67520
14. 6lin: Crystal Structure of Human Pdk2 Complexed with Gm10030
15. 6lil: Crystal Structure of Human Pdk2 Complexed with an Allosteric Inhibitor Compound 8c
16. 4mp2: Crystal Structure of Pyruvate Dehydrogenase Kinase Isoform 2 in Complex with Inhibitor Pa1
17. 4mp7: Crystal Structure of Pyruvate Dehydrogenase Kinase Isoform 2 in Complex with Inhibitor Pa7
18. 4mpc: Crystal Structure of Pyruvate Dehydrogenase Kinase Isoform 2 in Complex with Inhibitor Ps2
19. 4mpe: Crystal Structure of Pyruvate Dehydrogenase Kinase Isoform 2 in Complex with Inhibitor Ps8
20. 4mpn: Crystal Structure of Pyruvate Dehydrogenase Kinase Isoform 2 in Complex with Inhibitor Ps10
21. 4v25: Ver-246608, a Novel Pan-isoform Atp Competitive Inhibitor of Pyruvate Dehydrogenase Kinase, Disrupts Warburg Metabolism and Induces Context-dependent Cytostasis in Cancer Cells
22. 4v26: Ver-246608, a Novel Pan-isoform Atp Competitive Inhibitor of Pyruvate Dehydrogenase Kinase, Disrupts Warburg Metabolism and Induces Context-dependent Cytostasis in Cancer Cells
23. 5m4p: Application of Off-rate Screening in The Identification of Novel Pan- Isoform Inhibitors of Pyruvate Dehydrogenase Kinase
24. 5m4n: Application of Off-rate Screening in The Identification of Novel Pan- Isoform Inhibitors of Pyruvate Dehydrogenase Kinase
25. 5m4m: Application of Off-rate Screening in The Identification of Novel Pan- Isoform Inhibitors of Pyruvate Dehydrogenase Kinase
26. 5m4k: Application of Off-rate Screening in The Identification of Novel Pan- Isoform Inhibitors of Pyruvate Dehydrogenase Kinase
27. 5j71: Crystal Structure of Pyruvate Dehydrogenase Kinase Isoform 2 in Complex with Inhibitor Ps35
28. 5j6a: Crystal Structure of Pyruvate Dehydrogenase Kinase Isoform 2 in Complex with Inhibitor Ps46
29. 7ea0: Crystal Structure of Human Pyruvate Dehydrogenase Kinase 2 in Complex with Compound 1
30. 7eas: Crystal Structure of Human Pyruvate Dehydrogenase Kinase 2 in Complex with Compound 2
31. 7eat: Crystal Structure of Human Pyruvate Dehydrogenase Kinase 4 in Complex with Compound 1
32. 7ebb: Crystal Structure of Human Pyruvate Dehydrogenase Kinase 4 in Complex with Compound 2
33. 7ebg: Crystal Structure of Human Pyruvate Dehydrogenase Kinase 4 in Complex with Compound 7
34. 7ebh: Crystal Structure of Human Pyruvate Dehydrogenase Kinase 2 in Complex with Compound 13